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Dr. (8) Schlag, Peter M. Prof. Dr. (1) Schmitt, Clemens Prof. Dr. (6) Schmitt, Matthias Jürgen Dr. (1) Schöpe, Paul Curtis (2) Schreiber, Adrian PD Dr. med. (3) Schulz-Menger, Jeanette Prof. Dr. (26) Schütz, Anja Dr. (4) Schwarz, Roland Dr. (7) Schwedhelm, Carolina Dr. (1) Sczakiel, Henrike (2) Seidel, Franziska Dr. med. (3) Selbach, Matthias Prof. Dr. (4) Semenchenko, Egor (1) Serresi, Michela Dr. (1) Sholokh, Anastasiia (2) Siffrin, Volker (5) Sigal, Michael Dr. (11) Silvis, Casper (1) Simon, Katja Prof. Dr. (4) Smith, Janice (2) Solé Boldo, Llorenc Dr. rer. nat. 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Ahmed P. Ragunathan J. Shin S. Peter S. Kleissle M. Neuenschwander R. Schäfer J.P. von Kries G. Grüber P. Dröge 19. Oktober 2023 / Cell Chem Biol CLK2 and CLK4 are regulators of DNA damage-induced NF-κB targeted by novel small molecule inhibitors P. Mucka P. Lindemann B. Bosco M. Willenbrock S. Radetzki M. Neuenschwander C. Brischetto J.P. von Kries M. Nazaré C. Scheidereit 16. Oktober 2023 / eLife An unconventional gatekeeper mutation sensitizes inositol hexakisphosphate kinases to an allosteric inhibitor T. Aguirre S. Hostachy G.L. Dornan M. Neuenschwander C. Seyffarth V. Haucke A. Schütz J.P. von Kries D. Fiedler 10. Februar 2023 / Mol Syst Biol A single-cell RNA labeling strategy for measuring stress response upon tissue dissociation A. Neuschulz O. Bakina V. Badillo Lisakowski P. Olivares-Chauvet T. Conrad M. Gotthardt H. Kettenmann J.P. Junker 31. Januar 2023 / Cell Rep MDC1 maintains active elongation complexes of RNA polymerase II G. Pappas S.H.N. Munk K. Watanabe Q. Thomas Z. Gál H.H. Gram M.H. Lee D. Gómez-Cabello D.C. Kanellis P. Olivares-Chauvet D.H. Larsen L.H. Gregersen A. Maya-Mendoza P. Galanos J. Bartek 06. Februar 2023 / PLoS ONE Small molecule specifically inhibiting microglial nitric oxide release could become a potential treatment for neuroinflammation P. Jordan A. Costa E. Specker O. Popp A. Volkamer R. Piske T. Obrusnik S. Kleissle K. Stuke A. Rex M. Neuenschwander J.P. von Kries M. Nazare P. Mertins H. Kettenmann S.A. Wolf Januar 2023 / Nat Chem Biol Development of selective inhibitors of phosphatidylinositol 3-kinase C2α W.T. Lo H. Belabed M. Kücükdisli J. Metag Y. Roske P. Prokofeva Y. Ohashi A. Horatscheck D. Cirillo M. Krauss C. Schmied M. Neuenschwander J.P. von Kries G. Médard Be. Kuster O. Perisic R.L. Williams O. Daumke B. Payrastre S. Severin M. Nazaré V. Haucke 09. November 2023 / J Med Chem Structure-based design of xanthine-imidazopyridines and -imidazothiazoles as highly potent and in vivo efficacious tryptophan hydroxylase inhibitors E. Specker R. Wesolowski A. Schütz S. Matthes K. Mallow M. Wasinska-Kalwa L. Winkler A. Oder N. Alenina D. Pleimes J.P. von Kries U. Heinemann M. Bader M. Nazaré Dezember 2023 / Biomed Pharmacother Discovery of tetrazolo-pyridazine-based small molecules as inhibitors of MACC1-driven cancer metastasis S. Yan P.C. Schöpe J. Lewis K. Putzker U. Uhrig E. Specker J.P. von Kries P. Lindemann A. Omran H.E. Sanchez-Ibarra A. Unger M.L. Zischinsky B. Klebl W. Walther M. Nazaré D. Kobelt U. Stein Dezember 2023 / Dis Model Mech Neurofibromin 1 mutations impair the function of human induced pluripotent stem cell-derived microglia L.D. Kuhrt E. Motta N. Elmadany H. Weidling R. Fritsche-Guenther I.E. Efe O. Cobb J. Chatterjee L.G. Boggs M. Schnauß S. Diecke M. Semtner C. Anastasaki D.H. Gutmann H. 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August 2023 / FEBS Lett The FGFR inhibitor PD173074 binds to the C-terminus of oncofetal HMGA2 and modulates its DNA-binding and transcriptional activation functions S.M. Ahmed P. Ragunathan J. Shin S. Peter S. Kleissle M. Neuenschwander R. Schäfer J.P. von Kries G. Grüber P. Dröge
19. Oktober 2023 / Cell Chem Biol CLK2 and CLK4 are regulators of DNA damage-induced NF-κB targeted by novel small molecule inhibitors P. Mucka P. Lindemann B. Bosco M. Willenbrock S. Radetzki M. Neuenschwander C. Brischetto J.P. von Kries M. Nazaré C. Scheidereit
16. Oktober 2023 / eLife An unconventional gatekeeper mutation sensitizes inositol hexakisphosphate kinases to an allosteric inhibitor T. Aguirre S. Hostachy G.L. Dornan M. Neuenschwander C. Seyffarth V. Haucke A. Schütz J.P. von Kries D. Fiedler
10. Februar 2023 / Mol Syst Biol A single-cell RNA labeling strategy for measuring stress response upon tissue dissociation A. Neuschulz O. Bakina V. Badillo Lisakowski P. Olivares-Chauvet T. Conrad M. Gotthardt H. Kettenmann J.P. Junker
31. Januar 2023 / Cell Rep MDC1 maintains active elongation complexes of RNA polymerase II G. Pappas S.H.N. Munk K. Watanabe Q. Thomas Z. Gál H.H. Gram M.H. Lee D. Gómez-Cabello D.C. Kanellis P. Olivares-Chauvet D.H. Larsen L.H. Gregersen A. Maya-Mendoza P. Galanos J. Bartek
06. Februar 2023 / PLoS ONE Small molecule specifically inhibiting microglial nitric oxide release could become a potential treatment for neuroinflammation P. Jordan A. Costa E. Specker O. Popp A. Volkamer R. Piske T. Obrusnik S. Kleissle K. Stuke A. Rex M. Neuenschwander J.P. von Kries M. Nazare P. Mertins H. Kettenmann S.A. Wolf
Januar 2023 / Nat Chem Biol Development of selective inhibitors of phosphatidylinositol 3-kinase C2α W.T. Lo H. Belabed M. Kücükdisli J. Metag Y. Roske P. Prokofeva Y. Ohashi A. Horatscheck D. Cirillo M. Krauss C. Schmied M. Neuenschwander J.P. von Kries G. Médard Be. Kuster O. Perisic R.L. Williams O. Daumke B. Payrastre S. Severin M. Nazaré V. Haucke
09. November 2023 / J Med Chem Structure-based design of xanthine-imidazopyridines and -imidazothiazoles as highly potent and in vivo efficacious tryptophan hydroxylase inhibitors E. Specker R. Wesolowski A. Schütz S. Matthes K. Mallow M. Wasinska-Kalwa L. Winkler A. Oder N. Alenina D. Pleimes J.P. von Kries U. Heinemann M. Bader M. Nazaré
Dezember 2023 / Biomed Pharmacother Discovery of tetrazolo-pyridazine-based small molecules as inhibitors of MACC1-driven cancer metastasis S. Yan P.C. Schöpe J. Lewis K. Putzker U. Uhrig E. Specker J.P. von Kries P. Lindemann A. Omran H.E. Sanchez-Ibarra A. Unger M.L. Zischinsky B. Klebl W. Walther M. Nazaré D. Kobelt U. Stein
Dezember 2023 / Dis Model Mech Neurofibromin 1 mutations impair the function of human induced pluripotent stem cell-derived microglia L.D. Kuhrt E. Motta N. Elmadany H. Weidling R. Fritsche-Guenther I.E. Efe O. Cobb J. Chatterjee L.G. Boggs M. Schnauß S. Diecke M. Semtner C. Anastasaki D.H. Gutmann H. Kettenmann